Munyori: Janice Evans
Zuva Rekusika: 25 Chikunguru 2021
Gadziridza Zuva: 10 Chivabvu 2024
Anonim
Pharmacology of opicapone used for treatment of on-off phenomena seen with levodopa (New Drug 2020)
Vhidhiyo: Pharmacology of opicapone used for treatment of on-off phenomena seen with levodopa (New Drug 2020)

Zvemukati

Opicapone inoshandiswa pamwe chete nelevodopa uye carbidopa (Sinemet, Rytary) kurapa kupera-kwedosi 'kupfeka' zviratidzo zvehosha yaPasinson. Opicapone inhibitor yekatechol-O-methyltransferase (COMT). Opicapone inobatsira levodopa uye carbidopa kushanda zvirinani nekubvumira yakawanda yacho kusvika kuuropi, uko ine mhedzisiro yayo.

Opicapone inouya sekapuleti kutora nemuromo. Inowanzo kutorwa kamwe chete pazuva panguva yekurara uye inofanirwa kutorwa kanenge 1 awa zvisati zvaitika kana 1 awa mushure mekudya. Tevedza zvinongedzo pane yako tsamba yekunyora zvakanyatsonaka, uye bvunza chiremba wako kana wemishonga kuti atsanangure chero chikamu chausinganzwisise. Tora opicapone chaizvo sekurairwa. Usatore zvimwe kana zvishoma nezvayo kana kuitora kakawanda pane zvakatemwa nachiremba wako.

Opicapone inodzora chirwere chaPasinson asi haichirape. Ramba uchitora opicapone kunyangwe iwe uchinzwa zvakanaka. Usarega kutora opicapone usina kutaura nachiremba wako. Kana ukangoerekana warega kutora opicapone, unogona kukura chirwere chakakomba chinokonzera kupisa muviri, mhasuru dzakaomarara, kufamba kwemuviri zvisina kujairika, uye nyonganiso Chiremba wako angangoda kudzikisa dosi yako yeopicapone zvishoma uye nekuchinja madosi emimwe mishonga yako yechirwere chePasinson.


Kumbira wemishonga wako kana chiremba kopi yemashoko emugadziri wemurwere.

Mushonga uyu unogona kupihwa zvimwe zvinoshandiswa; bvunza chiremba wako kana wemishonga kuti uwane rumwe ruzivo.

Usati watora opicapone,

  • udza chiremba wako uye wemishonga kana uri weergoria kune opicapone, chero mimwe mishonga, kana chero chinhu chinowanikwa muopicapone capusules. Kumbira wako wemishonga kuti uwane runyorwa rwezvigadzirwa.
  • udza chiremba wako kana uri kutora isocarboxazid (Marplan), phenelzine (Nardil) kana tranylcypromine (Parnate) kana kuti warega kuatora mumavhiki maviri apfuura. Chiremba wako angangokuudza kuti usatora opicapone.
  • udza chiremba wako uye wemishonga kuti ndeipi imwe mishonga yekunyorera uye isina kunyoreswa, mavitamini, zvinowedzera zvinovaka muviri, uye mishonga yemakwenzi yauri kutora kana kuronga kutora.Ive neshuwa yekutaura chero eanotevera: mishonga yekukwira kweropa, mishonga inokonzeresa kukotsira, dobutamine, epinephrine (Epipen, Primatine Mist, vamwe), mishonga yekuzorodza, mapiritsi ekurara, uye tranquilizers. Chiremba wako angangoda kushandura madosi emishonga yako kana kukutarisisa nokungwarira mhedzisiro. Mimwe mishonga yakawanda inogona zvakare kubatana neopicapone, saka ive shuwa kuudza chiremba wako nezve yese mishonga yauri kutora, kunyangwe iyo isingaonekwe pane ino runyorwa.
  • udza chiremba wako kana iwe uine pheochromocytoma kana paraganglioma (mamota pane kana kutenderedza gland diki padyo neitsvo). Chiremba wako angangokuudza kuti usatora opicapone.
  • udza chiremba wako kana wakambove nehope dzemasikati dzisingatarisirwi kana chirwere chekurara, dyskinesia (isingadzorwe kufamba kamwe kamwe), chirwere chepfungwa (chirwere chepfungwa chinokonzera kufunga zvisina kujairika kana kufunga), kana chiropa kana chirwere cheitsvo.
  • udza chiremba wako kana iwe uri nepamuviri, ronga kuve nepamuviri, kana uri kuyamwisa. Kana iwe ukava nepamuviri uchitora opicapone, fonera chiremba wako.
  • kana uri kuvhiyiwa, kusanganisira kuvhiya mazino, udza chiremba kana chiremba wemazino kuti urikutora opicapone.
  • iwe unofanirwa kuziva kuti opicapone inogona kukuwisira iwe kana inogona kukukonzera iwe kukotsira kamwe kamwe panguva yemabasa ako ezuva nezuva. Iwe unogona kusanzwa kukotsira kana kuve nechero imwe zviratidzo zvekuyambira usati warara kamwe kamwe. Usafambisa mota, kushandisa michina, kushanda pakakwirira, kana kutora chikamu mune zvinogona kuita njodzi zviitiko pakutanga kwekurapwa kwako kusvika iwe waziva kuti mushonga unokubata sei. Kana iwe ukangoerekana warara iwe paunenge uchiita chimwe chinhu senge kutarisa terevhizheni, kutaura, kudya, kana kukwira mumotokari, kana kana iwe ukanyanya kukotsira, kunyanya panguva yemasikati, fonera chiremba wako. Usafambisa, shanda munzvimbo dzakakwirira, kana kushandisa michina kusvikira wataura nachiremba wako.
  • rangarira kuti doro rinogona kuwedzera kuhope dzinokonzerwa nemushonga uyu. Udza chiremba wako kana uchigara uchinwa zvinwiwa zvinodhaka.
  • iwe unofanirwa kuziva kuti vamwe vanhu vakatora mishonga senge opicapone vakagadzira matambudziko nyowani kana akawedzera ekubhejera kana zvimwe zvinokurudzira zvakanyanya kana hunhu hwaive hwekumanikidza kana husina kujairika kwavari, sekuwedzera kwekushuva kwepabonde kana maitiro. Iko hakuna ruzivo rwakaringana kutaura kuti vanhu vakagadzira matambudziko aya nekuti ivo vakatora mushonga kana nekuda kwezvimwe zvikonzero. Fonera chiremba wako kana iwe uine shungu yekubheja iyo yakaoma kudzora, iwe une zvakakomba kukurudzira, kana iwe uri kutadza kudzora maitiro ako. Udza nhengo dzemhuri yako nezve njodzi iyi kuitira kuti vafonere chiremba kunyangwe iwe usinga zive kuti kubhejera kwako kana zvimwe zvinokuchidzira zvakanyanya kana maitiro asina kujairika rave dambudziko.
  • iwe unofanirwa kuziva kuti opicapone inogona kukonzeresa dzungu, huremu husina musoro, uye kupera simba paunosimuka nekukurumidza kubva panzvimbo yekunyepa. Izvi zvinowanzoitika kana iwe ukatanga kutora opicapone. Kuti udzivise dambudziko iri, simuka pamubhedha zvishoma nezvishoma, uchizorora tsoka dzako pasi kwemaminetsi mashoma usati wasimuka.

Kunze kwekunge chiremba wako akakuudza neimwe nzira, ramba uchidya zvakajairika.


Iwe unofanirwa kusvetuka iro rakarasika dosi. Tora dosi yako yenguva dzose panguva yako inotevera yekurara. Usapeta kaviri muyero unotevera kuti uwane dhosi rakarasika.

Opicapone inogona kukonzera mhedzisiro. Udza chiremba wako kana chimwe chezviratidzo izvi chakanyanya kana kuti chisingaendi:

  • kuvimbiswa
  • muromo wakaoma
  • kunetseka kurara kana kuramba wakarara
  • dzungu
  • kuonda
  • kufamba zvisina kujairika kana kusadzora kwemuviri

Mimwe mhedzisiro inogona kuve yakakomba. Kana iwe uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchinge uchida kurapwa,

  • kufungidzira (kuona zvinhu kana kunzwa manzwi zvisipo)
  • kunyengera (kuva nemafungiro asinganzwisisike kana zvitendero zvisina hwaro muzvokwadi)
  • hunhu hwehasha
  • kufenda

Opicapone inogona kukonzera mamwe mhedzisiro. Fonera chiremba wako kana uine chero matambudziko asina kujairika uchitora mushonga uyu.

Kana iwe ukawana chakakomba mhedzisiro, iwe kana chiremba wako ungatumira chirevo kuchirongwa cheKudya neDrug Administration's (FDA) MedWatch Yakashata Chiitiko Chirongwa online (http://www.fda.gov/Safety/MedWatch) kana nefoni ( 1-800-332-1088).


Chengetedza iyi mishonga mumudziyo iyo yakauya mukati, yakasungwa yakavharwa, uye isingasvike kune vana. Zvichengetedze pane tembiricha yemukati uye kure nechiedza, kupisa kwakanyanya uye hunyoro (kwete muchimbuzi).

Izvo zvakakosha kuti chengetedza mishonga yese isingaonekwe uye kusvika kwevana semidziyo yakawanda (senge vhiki nevhiki mapiritsi epfungwa uye ayo emadonhwe eziso, makirimu, zvigamba, uye inhalers) hazvirambe vana uye vana vadiki vanogona kuvhura zviri nyore. Kuchengetedza vana vadiki kubva kune chepfu, gara wakavharira makapu ekuchengetedza uye nekukurumidza isa mishonga munzvimbo yakachengeteka - imwe iri kumusoro uye kure uye kubva kwavari uye kusvika. http://www.upandaway.org

Mishonga isingadiwe inofanirwa kuraswa nenzira dzakakosha kuona kuti zvipfuyo, vana, nevamwe vanhu havagone kuzvidya. Nekudaro, iwe haufanire kuburitsa uyu mushonga pasi pechimbuzi. Panzvimbo iyoyo, nzira yakanakisa yekurasa mishonga yako ndeyekurapa-kudzosa chirongwa. Taura nachiremba wako kana kuti taura nedhipatimendi rako remarara / rekudzokorora kuti udzidze nezve zvirongwa zvekudzosa munharaunda yako. Ona iyo FDA's Safe Disposal yeMedicine webhusaiti (http://goo.gl/c4Rm4p) kuti uwane rumwe ruzivo kana iwe usina mukana wekutora-kudzoka chirongwa.

Kana zvikaitika zvekudarika, fonera iyo chepfu yekudzora rubatsiro pa1-800-222-1222. Ruzivo rwunowanikwawo online pa https://www.poisonhelp.org/help. Kana munhu akabatwa akadonha, akabatwa nepfari, achinetseka kufema, kana kutadza kumutswa, pakarepo danaidza mabasa ekukurumidzira pa911.

Chengetedza zvese zvakagadzwa nachiremba wako.

Usarega mumwe munhu achitora mushonga wako. Kumbira wemishonga wako chero mibvunzo yauinayo nezvekuzadza tsamba yako.

Izvo zvakakosha kuti iwe uchengete yakanyorwa rondedzero yeese emushonga uye asiri ekunyora (pamusoro-e-pikisheni) mishonga yauri kutora, pamwe nezvimwe zvigadzirwa zvakaita sevhitamini, zvicherwa, kana zvimwe zvekuwedzera zvekudya. Iwe unofanirwa kuuya nerondedzero iyi iwe nguva imwe neimwe paunoshanyira chiremba kana kana iwe uchigamuchirwa kuchipatara. Izvo zvakare zvakakosha ruzivo kutakura newe kana zvikaitika zvechimbi-chimbi.

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